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Bioorganic & Medicinal Chemistry Letters

  1. Electron affinity of tricyclic, bicyclic, and monocyclic compounds containing cyanoenones correlates with their potency as inducers of a cytoprotective enzyme

    Bensasson, R. V., Dinkova-Kostova, A. T., Zheng, S., Saito, A., Li, W., Zoete, V. & Honda, T. 1 Sep 2016 In : Bioorganic & Medicinal Chemistry Letters. 26, 17, p. 4345-4349 5 p.

    Research output: Contribution to journalArticle

  2. Synthesis and structure-activity relationships of a novel series of pyrimidines as potent inhibitors of TBK1/IKKε kinases

    McIver, E. G., Bryans, J., Birchall, K., Chugh, J., Drake, T., Lewis, S. J., Osborne, J., Smiljanic-Hurley, E., Tsang, W., Kamal, A., Levy, A., Newman, M., Taylor, D., Arthur, J. S. C., Clark, K. & Cohen, P. Dec 2012 In : Bioorganic & Medicinal Chemistry Letters. 22, 23, p. 7169-7173 5 p.

    Research output: Contribution to journalArticle

  3. Characterization of TAE684 as a potent LRRK2 kinase inhibitor

    Zhang, J., Deng, X., Choi, H. G., Alessi, D. R. & Gray, N. S. 1 Mar 2012 In : Bioorganic & Medicinal Chemistry Letters. 22, 5, p. 1864-1869 6 p.

    Research output: Contribution to journalArticle

  4. Inhibitors of human histone deacetylase with potent activity against the African trypanosome Trypanosoma brucei

    Kelly, J. M., Taylor, M. C., Horn, D., Loza, E., Kalvinsh, I. & Bjorkling, F. 1 Mar 2012 In : Bioorganic & Medicinal Chemistry Letters. 22, 5, p. 1886-1890 5 p.

    Research output: Contribution to journalArticle

  5. GSK2578215A: a potent and highly selective 2-arylmethyloxy-5-substitutent-N-arylbenzamide LRRK2 kinase inhibitor

    Reith, A. D., Bamborough, P., Jandu, K., Andreotti, D., Mensah, L., Dossang, P., Choi, H. G., Deng, X., Zhang, J., Alessi, D. R. & Gray, N. S. 2012 In : Bioorganic & Medicinal Chemistry Letters. 22, 17, p. 5625-5629 5 p.

    Research output: Contribution to journalArticle

  6. High-affinity fluorescent ligands for the 5-HT3 receptor

    Simonin, J., Vernekar, S. K. V., Thompson, A. J., Hothersall, J. D., Connolly, C. N., Lummis, S. C. R. & Lochner, M. 2012 In : Bioorganic & Medicinal Chemistry Letters. 22, 2, p. 1151-1155 5 p.

    Research output: Contribution to journalArticle

  7. Synthesis and biological evaluation of 1-[2-cyano-3,12-dioxooleana-1,9(11)-dien-28-oyl]-4-ethynylimidazole. A novel and highly potent anti-inflammatory and cytoprotective agent

    Honda, T., Dinkova-Kostova, A. T., David, E., Padegimas, E. M., Sundararajan, C., Visnick, M., Bumeister, R. & Wigley, W. C. 15 Apr 2011 In : Bioorganic & Medicinal Chemistry Letters. 21, 8, p. 2188-2191 4 p.

    Research output: Contribution to journalArticle

  8. Selective delivery of 2-hydroxy APA to Trypanosoma brucei using the melamine motif

    Klee, N., Wong, P. E., Baragana, B., El Mazouni, F., Phillips, M. A., Barrett, M. P. & Gilbert, I. H. 1 Aug 2010 In : Bioorganic & Medicinal Chemistry Letters. 20, 15, p. 4364-4366 3 p.

    Research output: Contribution to journalArticle

  9. Structure-based optimization of potent PDK1 inhibitors

    Angiolini, M., Banfi, P., Casale, E., Casuscelli, F., Fiorelli, C., Saccardo, M. B., Silvagni, M. & Zuccotto, F. 15 Jul 2010 In : Bioorganic & Medicinal Chemistry Letters. 20, 14, p. 4095-4099 5 p.

    Research output: Contribution to journalArticle

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