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Bioorganic & Medicinal Chemistry Letters

  1. Synthesis and structure-activity relationships of a novel series of pyrimidines as potent inhibitors of TBK1/IKKε kinases

    McIver, E. G., Bryans, J., Birchall, K., Chugh, J., Drake, T., Lewis, S. J., Osborne, J., Smiljanic-Hurley, E., Tsang, W., Kamal, A., Levy, A., Newman, M., Taylor, D., Arthur, J. S. C., Clark, K. & Cohen, P. Dec 2012 In : Bioorganic & Medicinal Chemistry Letters. 22, 23, p. 7169-7173 5 p.

    Research output: Contribution to journalArticle

  2. Characterization of TAE684 as a potent LRRK2 kinase inhibitor

    Zhang, J., Deng, X., Choi, H. G., Alessi, D. R. & Gray, N. S. 1 Mar 2012 In : Bioorganic & Medicinal Chemistry Letters. 22, 5, p. 1864-1869 6 p.

    Research output: Contribution to journalArticle

  3. Inhibitors of human histone deacetylase with potent activity against the African trypanosome Trypanosoma brucei

    Kelly, J. M., Taylor, M. C., Horn, D., Loza, E., Kalvinsh, I. & Bjorkling, F. 1 Mar 2012 In : Bioorganic & Medicinal Chemistry Letters. 22, 5, p. 1886-1890 5 p.

    Research output: Contribution to journalArticle

  4. GSK2578215A: a potent and highly selective 2-arylmethyloxy-5-substitutent-N-arylbenzamide LRRK2 kinase inhibitor

    Reith, A. D., Bamborough, P., Jandu, K., Andreotti, D., Mensah, L., Dossang, P., Choi, H. G., Deng, X., Zhang, J., Alessi, D. R. & Gray, N. S. 2012 In : Bioorganic & Medicinal Chemistry Letters. 22, 17, p. 5625-5629 5 p.

    Research output: Contribution to journalArticle

  5. High-affinity fluorescent ligands for the 5-HT3 receptor

    Simonin, J., Vernekar, S. K. V., Thompson, A. J., Hothersall, J. D., Connolly, C. N., Lummis, S. C. R. & Lochner, M. 2012 In : Bioorganic & Medicinal Chemistry Letters. 22, 2, p. 1151-1155 5 p.

    Research output: Contribution to journalArticle

  6. Synthesis and biological evaluation of 1-[2-cyano-3,12-dioxooleana-1,9(11)-dien-28-oyl]-4-ethynylimidazole. A novel and highly potent anti-inflammatory and cytoprotective agent

    Honda, T., Dinkova-Kostova, A. T., David, E., Padegimas, E. M., Sundararajan, C., Visnick, M., Bumeister, R. & Wigley, W. C. 15 Apr 2011 In : Bioorganic & Medicinal Chemistry Letters. 21, 8, p. 2188-2191 4 p.

    Research output: Contribution to journalArticle

  7. Selective delivery of 2-hydroxy APA to Trypanosoma brucei using the melamine motif

    Klee, N., Wong, P. E., Baragana, B., El Mazouni, F., Phillips, M. A., Barrett, M. P. & Gilbert, I. H. 1 Aug 2010 In : Bioorganic & Medicinal Chemistry Letters. 20, 15, p. 4364-4366 3 p.

    Research output: Contribution to journalArticle

  8. The identification a novel, selective, non-steroidal, functional glucocorticoid receptor antagonist

    Rimland, J., Dunne, A., Hunjan, S. S., Sasse, R., Uings, I., Montanari, D., Caivano, M., Shah, P., Standing, D., Gray, D., Brown, D., Cairns, W., Trump, R., Smith, P. W., Bertheleme, N., D'Alessandro, P., Gul, S., Vimal, M., Smith, D. N. & Watson, S. P. Apr 2010 In : Bioorganic & Medicinal Chemistry Letters. 20, 7, p. 2340-3 4 p.

    Research output: Contribution to journalArticle

  9. Synthesis of 3-alkyl naphthalenes as novel estrogen receptor ligands

    Fang, J., Akwabi-Ameyaw, A., Britton, J. E., Katamreddy, S. R., Navas III, F., Miller, A. B., Williams, S. P., Gray, D. W., Orband-Miller, L. A., Shearin, J. & Heyer, D. 15 Sep 2008 In : Bioorganic & Medicinal Chemistry Letters. 18, 18, p. 5075-5077 3 p.

    Research output: Contribution to journalArticle

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