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Journal of Medicinal Chemistry

  1. Allosteric targeting of the Fanconi anemia ubiquitin-conjugating enzyme Ube2T by fragment screening

    Morreale, F., Bortoluzzi, A., Chaugule, V., Arkinson, C., Walden, H. & Ciulli, A. 11 May 2017 In : Journal of Medicinal Chemistry. 60, 9, p. 4093-4098 6 p.

    Research output: Contribution to journalArticle

  2. Kinetin Riboside and Its ProTides Activate the Parkinson’s Disease Associated PTEN-Induced Putative Kinase 1 (PINK1) Independent of Mitochondrial Depolarization

    Osgerby, L., Lai, Y-C., Thornton, P. J., Amalfitano, J., Le Duff, C. S., Jabeen, I., Kadri, H., Miccoli, A., Tucker, J. H. R., Muqit, M. M. K. & Mehellou, Y. 27 Apr 2017 In : Journal of Medicinal Chemistry. 60, 8, p. 3518-3524 7 p.

    Research output: Contribution to journalArticle

  3. Targeting Bacillosamine Biosynthesis in Bacterial Pathogens: Development of Inhibitors to a Bacterial Amino-Sugar Acetyltransferase from Campylobacter jejuni

    De Schutter, J. W., Morrison, J. P., Morrison, M. J., Ciulli, A. & Imperiali, B. 9 Mar 2017 In : Journal of Medicinal Chemistry. 60, 5, p. 2099-2118 20 p.

    Research output: Contribution to journalArticle

  4. Discovery of a quinoline-4-carboxamide derivative with a novel mechanism of action, multistage antimalarial activity, and potent in vivo efficacy

    Gilbert, I. H. & 26 others Baragaña, B., Norcross, N. R., Wilson, C., Porzelle, A., Hallyburton, I., Grimaldi, R., Osuna-Cabello, M., Norval, S., Riley, J., Stojanovski, L., Simeons, F. R. C., Wyatt, P. G., Delves, M. J., Meister, S., Duffy, S., Avery, V. M., Winzeler, E. A., Sinden, R. E., Wittlin, S., Frearson, J. A., Gray, D. W., Fairlamb, A. H., Waterson, D., Campbell, S. F., Willis, P. & Read, K. D. 10 Nov 2016 In : Journal of Medicinal Chemistry. 59, 21, p. 9672-9685 14 p.

    Research output: Contribution to journalArticle

  5. Hit-to-Lead Optimization of a Novel Class of Potent, Broad-Spectrum Trypanosomacides

    Thomas, J. & 25 others Russell, S., Rahmani, R., Jones, A. J., Newson, H. L., Neilde, K., Cotillo, I., Rahmani Khajouei, M., Ferrins, L., Qureishi, S., Nguyen, N., Martinez-Martinez, M. S., Weaver, D. F., Kaiser, M., Riley, J., De Rycker, M., Read, K. D., Flematti, G. R., Ryan, E., Tanghe, S., Rodriguez, A., Charman, S. A., Kessler, A., Avery, V. M., Baell, J. B. & Piggott, M. J. 10 Nov 2016 In : Journal of Medicinal Chemistry. 59, 21, p. 9686-9720 35 p.

    Research output: Contribution to journalArticle

  6. From Companion Diagnostics to Theranostics: A New Avenue for Alzheimer's Disease?

    Bolognesi, M. L., Gandini, A., Prati, F. & Uliassi, E. 8 Sep 2016 In : Journal of Medicinal Chemistry. 59, 17, p. 7759-7770 12 p.

    Research output: Contribution to journalReview article

  7. Trisubstituted Pyrimidines as Efficacious and Fast-acting Antimalarials

    Gilbert, I. H. & 29 others Norcross, N. R., Baragana, B., Wilson, C., Hallyburton, I., Osuna-Cabello, M., Norval, S., Riley, J., Stojanovski, L., Simeons, F. R. C., Porzelle, A., Grimaldi, R., Wittlin, S., Duffy, S., Avery, V. M., Meister, S., Sanz, L., Jimenez-Diaz, B., Angulo-Barturen, I., Ferrer, S., Santos Marinez, M., Javier Gamo, F., Frearson, J. A., Gray, D. W., Fairlamb, A. H., Winzeler, E. A., Waterson, D., Campbell, S. F., Willis, P. & Read, K. D. 14 Jul 2016 In : Journal of Medicinal Chemistry. 59, 13, p. 6101-6120 20 p.

    Research output: Contribution to journalArticle

  8. 4-Acyl Pyrrole Derivatives Yield Novel Vectors for Designing Inhibitors of the Acetyl-Lysine Recognition Site of BRD4(1)

    Hügle, M., Lucas, X., Weitzel, G., Ostrovskyi, D., Breit, B., Gerhardt, S., Einsle, O., Günther, S. & Wohlwend, D. 25 Feb 2016 In : Journal of Medicinal Chemistry. 59, 4, p. 1518-1530 13 p.

    Research output: Contribution to journalArticle

  9. New synthetic routes to Triazolo-benzodiazepine analogues: expanding the scope of the bump-and-hole approach for selective Bromo and Extra-Terminal (BET) bromodomain inhibition

    Baud, M. G. J., Lin-Shiao, E., Zengerle, M., Tallant, C. & Ciulli, A. 25 Feb 2016 In : Journal of Medicinal Chemistry. 59, 4, p. 1492-1500 9 p.

    Research output: Contribution to journalArticle

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