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Journal of Medicinal Chemistry

  1. Allosteric targeting of the Fanconi anemia ubiquitin-conjugating enzyme Ube2T by fragment screening

    Morreale, F., Bortoluzzi, A., Chaugule, V., Arkinson, C., Walden, H. & Ciulli, A. 11 May 2017 In : Journal of Medicinal Chemistry. 60, 9, p. 4093-4098 6 p.

    Research output: Contribution to journalArticle

  2. Kinetin Riboside and Its ProTides Activate the Parkinson’s Disease Associated PTEN-Induced Putative Kinase 1 (PINK1) Independent of Mitochondrial Depolarization

    Osgerby, L., Lai, Y-C., Thornton, P. J., Amalfitano, J., Le Duff, C. S., Jabeen, I., Kadri, H., Miccoli, A., Tucker, J. H. R., Muqit, M. M. K. & Mehellou, Y. 27 Apr 2017 In : Journal of Medicinal Chemistry. 60, 8, p. 3518-3524 7 p.

    Research output: Contribution to journalArticle

  3. Targeting Bacillosamine Biosynthesis in Bacterial Pathogens: Development of Inhibitors to a Bacterial Amino-Sugar Acetyltransferase from Campylobacter jejuni

    De Schutter, J. W., Morrison, J. P., Morrison, M. J., Ciulli, A. & Imperiali, B. 9 Mar 2017 In : Journal of Medicinal Chemistry. 60, 5, p. 2099-2118 20 p.

    Research output: Contribution to journalArticle

  4. Discovery of a quinoline-4-carboxamide derivative with a novel mechanism of action, multistage antimalarial activity, and potent in vivo efficacy

    Baragaña, B. , Norcross, N. R. , Wilson, C. , Porzelle, A. , Hallyburton, I. , Grimaldi, R. , Osuna-Cabello, M. , Norval, S. , Riley, J. , Stojanovski, L. , Simeons, F. R. C. , Wyatt, P. G. , Delves, M. J. , Meister, S. , Duffy, S. , Avery, V. M. , Winzeler, E. A. , Sinden, R. E. , Wittlin, S. , Frearson, J. A. & 7 others Gray, D. W., Fairlamb, A. H., Waterson, D., Campbell, S. F., Willis, P., Read, K. D. & Gilbert, I. H. 10 Nov 2016 In : Journal of Medicinal Chemistry. 59, 21, p. 9672-9685 14 p.

    Research output: Contribution to journalArticle

  5. Hit-to-Lead Optimization of a Novel Class of Potent, Broad-Spectrum Trypanosomacides

    Russell, S. , Rahmani, R. , Jones, A. J. , Newson, H. L. , Neilde, K. , Cotillo, I. , Rahmani Khajouei, M. , Ferrins, L. , Qureishi, S. , Nguyen, N. , Martinez-Martinez, M. S. , Weaver, D. F. , Kaiser, M. , Riley, J. , Thomas, J. , De Rycker, M. , Read, K. D. , Flematti, G. R. , Ryan, E. , Tanghe, S. & 6 others Rodriguez, A., Charman, S. A., Kessler, A., Avery, V. M., Baell, J. B. & Piggott, M. J. 10 Nov 2016 In : Journal of Medicinal Chemistry. 59, 21, p. 9686-9720 35 p.

    Research output: Contribution to journalArticle

  6. From Companion Diagnostics to Theranostics: A New Avenue for Alzheimer's Disease?

    Bolognesi, M. L., Gandini, A., Prati, F. & Uliassi, E. 8 Sep 2016 In : Journal of Medicinal Chemistry. 59, 17, p. 7759-7770 12 p.

    Research output: Contribution to journalReview article

  7. Trisubstituted Pyrimidines as Efficacious and Fast-acting Antimalarials

    Norcross, N. R. , Baragana, B. , Wilson, C. , Hallyburton, I. , Osuna-Cabello, M. , Norval, S. , Riley, J. , Stojanovski, L. , Simeons, F. R. C. , Porzelle, A. , Grimaldi, R. , Wittlin, S. , Duffy, S. , Avery, V. M. , Meister, S. , Sanz, L. , Jimenez-Diaz, B. , Angulo-Barturen, I. , Ferrer, S. , Santos Marinez, M. & 10 others Javier Gamo, F., Frearson, J. A., Gray, D. W., Fairlamb, A. H., Winzeler, E. A., Waterson, D., Campbell, S. F., Willis, P., Read, K. D. & Gilbert, I. H. 14 Jul 2016 In : Journal of Medicinal Chemistry. 59, 13, p. 6101-6120 20 p.

    Research output: Contribution to journalArticle

  8. 4-Acyl Pyrrole Derivatives Yield Novel Vectors for Designing Inhibitors of the Acetyl-Lysine Recognition Site of BRD4(1)

    Hügle, M., Lucas, X., Weitzel, G., Ostrovskyi, D., Breit, B., Gerhardt, S., Einsle, O., Günther, S. & Wohlwend, D. 25 Feb 2016 In : Journal of Medicinal Chemistry. 59, 4, p. 1518-1530 13 p.

    Research output: Contribution to journalArticle

  9. New synthetic routes to Triazolo-benzodiazepine analogues: expanding the scope of the bump-and-hole approach for selective Bromo and Extra-Terminal (BET) bromodomain inhibition

    Baud, M. G. J., Lin-Shiao, E., Zengerle, M., Tallant, C. & Ciulli, A. 25 Feb 2016 In : Journal of Medicinal Chemistry. 59, 4, p. 1492-1500 9 p.

    Research output: Contribution to journalArticle

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