Discovery - University of Dundee - Online Publications

Library & Learning Centre

Journal of Medicinal Chemistry

1 - 10 out of 36Page size: 10
Sort by: Publication year
  1. Targeting low-druggability bromodomains: fragment based screening and inhibitor design against the BAZ2B bromodomain

    Ferguson, F. M., Fedorov, O., Chaikuad, A., Philpott, M., Muniz, J. R. C., Felletar, I., von Delft, F., Heightman, T., Knapp, S., Abell, C. & Ciulli, A. Dec 2013 In : Journal of Medicinal Chemistry. 56, 24, p. 10183-10187 5 p.

    Research output: Contribution to journalArticle

  2. X-ray crystal structure of ERK5 (MAPK7) in complex with a specific inhibitor

    Elkins, J. M., Wang, J., Deng, X., Pattison, M. J., Arthur, J. S. C., Erazo, T., Gomez, N., Lizcano, J. M., Gray, N. S. & Knapp, S. 13 Jun 2013 In : Journal of Medicinal Chemistry. 56, 11, p. 4413-4421 9 p.

    Research output: Contribution to journalArticle

  3. Discovery and structure-activity relationships of pyrrolone antimalarials

    Murugesan, D., Mital, A., Kaiser, M., Shackleford, D. M., Morizzi, J., Katneni, K., Campbell, M., Hudson, A., Charman, S. A., Yeates, C. & Gilbert, I. H. 2013 In : Journal of Medicinal Chemistry. 56, 7, p. 2975-2990 16 p.

    Research output: Contribution to journalArticle

  4. Drug discovery for neglected diseases: molecular target-based and phenotypic approaches

    Gilbert, I. H. 2013 In : Journal of Medicinal Chemistry. 56, 20, p. 7719-7726 8 p.

    Research output: Contribution to journalArticle

  5. Synthesis, chemical reactivity as Michael acceptors, and biological potency of monocyclic cyanoenones, novel and highly potent anti-inflammatory and cytoprotective agents

    Zheng, S., Laxmi, Y. R. S., David, E., Dinkova-Kostova, A. T., Shiavoni, K. H., Ren, Y., Zheng, Y., Trevino, I., Bumeister, R., Ojima, I., Wigley, W. C., Bliska, J. B., Mierke, D. F. & Honda, T. 24 May 2012 In : Journal of Medicinal Chemistry. 55, 10, p. 4837-4846 10 p.

    Research output: Contribution to journalArticle

  6. Discovery of a Novel Class of Orally Active Trypanocidal N-Myristoyltransferase Inhibitors

    Brand, S., Cleghorn, L. A. T., McElroy, S. P., Robinson, D. A., Smith, V. C., Hallyburton, I., Harrison, J. R., Norcross, N. R., Spinks, D., Bayliss, T., Norval, S., Stojanovski, L., Torrie, L. S., Frearson, J. A., Brenk, R., Fairlamb, A. H., Ferguson, M. A. J., Read, K. D., Wyatt, P. G. & Gilbert, I. H. 12 Jan 2012 In : Journal of Medicinal Chemistry. 55, 1, p. 140-152 13 p.

    Research output: Contribution to journalArticle

  7. Synthesis and Evaluation of α-Thymidine Analogues as Novel Antimalarials

    Cui, H., Carrero-Lérida, J., Silva, A. P. G., Whittingham, J. L., Brannigan, J. A., Ruiz-Pérez, L. M., Read, K. D., Wilson, K. S., González-Pacanowska, D. & Gilbert, I. H. 2012 In : Journal of Medicinal Chemistry. 55, 24, p. 10948-57 10 p.

    Research output: Contribution to journalArticle

  8. Dihydroquinazolines as a Novel Class of Trypanosoma brucei Trypanothione Reductase Inhibitors: Discovery, Synthesis, and Characterization of their Binding Mode by Protein Crystallography

    Patterson, S., Alphey, M. S., Jones, D. C., Shanks, E. J., Street, I. P., Frearson, J. A., Wyatt, P. G., Gilbert, I. H. & Fairlamb, A. H. 13 Oct 2011 In : Journal of Medicinal Chemistry. 54, 19, p. 6514-6530 17 p.

    Research output: Contribution to journalArticle

  9. 6-(3,4-dichlorophenyl)-1-[(methyloxy)methyl]-3-azabicyclo[4.1.0]heptane: a new potent and selective triple reuptake inhibitor

    Micheli, F. , Cavanni, P. , Andreotti, D. , Arban, R. , Benedetti, R. , Bertani, B. , Bettati, M. , Bettelini, L. , Bonanomi, G. , Braggio, S. , Carletti, R. , Checchia, A. , Corsi, M. , Fazzolari, E. , Fontana, S. , Marchioro, C. , Merlo-Pich, E. , Negri, M. , Oliosi, B. , Ratti, E. & 11 others Read, K. D., Roscic, M., Sartori, I., Spada, S., Tedesco, G., Tarsi, L., Terreni, S., Visentini, F., Zocchi, A., Zonzini, L. & Di Fabio, R. 8 Jul 2010 In : Journal of Medicinal Chemistry. 53, 13, p. 4989-5001 13 p.

    Research output: Contribution to journalArticle

Previous 1 2 3 4 Next

Library & Learning Centre

Contact | Accessibility | Policy