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High-affinity fluorescent ligands for the 5-HT3 receptor

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High-affinity fluorescent ligands for the 5-HT3 receptor. / Simonin, Jonathan; Vernekar, Sanjeev Kumar V.; Thompson, Andrew J.; Hothersall, J. Daniel; Connolly, Christopher N.; Lummis, Sarah C. R.; Lochner, Martin.

In: Bioorganic & Medicinal Chemistry Letters, Vol. 22, No. 2, 2012, p. 1151-1155.

Research output: Contribution to journalArticle

Harvard

Simonin, J, Vernekar, SKV, Thompson, AJ, Hothersall, JD, Connolly, CN, Lummis, SCR & Lochner, M 2012, 'High-affinity fluorescent ligands for the 5-HT3 receptor' Bioorganic & Medicinal Chemistry Letters, vol 22, no. 2, pp. 1151-1155.

APA

Simonin, J., Vernekar, S. K. V., Thompson, A. J., Hothersall, J. D., Connolly, C. N., Lummis, S. C. R., & Lochner, M. (2012). High-affinity fluorescent ligands for the 5-HT3 receptor. Bioorganic & Medicinal Chemistry Letters, 22(2), 1151-1155doi: 10.1016/j.bmcl.2011.11.097

Vancouver

Simonin J, Vernekar SKV, Thompson AJ, Hothersall JD, Connolly CN, Lummis SCR et al. High-affinity fluorescent ligands for the 5-HT3 receptor. Bioorganic & Medicinal Chemistry Letters. 2012;22(2):1151-1155.

Author

Simonin, Jonathan; Vernekar, Sanjeev Kumar V.; Thompson, Andrew J.; Hothersall, J. Daniel; Connolly, Christopher N.; Lummis, Sarah C. R.; Lochner, Martin / High-affinity fluorescent ligands for the 5-HT3 receptor.

In: Bioorganic & Medicinal Chemistry Letters, Vol. 22, No. 2, 2012, p. 1151-1155.

Research output: Contribution to journalArticle

Bibtex - Download

@article{e5adf219b8154118b6277490a193f007,
title = "High-affinity fluorescent ligands for the 5-HT3 receptor",
author = "Jonathan Simonin and Vernekar, {Sanjeev Kumar V.} and Thompson, {Andrew J.} and Hothersall, {J. Daniel} and Connolly, {Christopher N.} and Lummis, {Sarah C. R.} and Martin Lochner",
note = "Copyright © 2011 Elsevier Ltd. All rights reserved.",
year = "2012",
volume = "22",
number = "2",
pages = "1151--1155",
journal = "Bioorganic & Medicinal Chemistry Letters",
issn = "0960-894X",

}

RIS (suitable for import to EndNote) - Download

TY - JOUR

T1 - High-affinity fluorescent ligands for the 5-HT3 receptor

A1 - Simonin,Jonathan

A1 - Vernekar,Sanjeev Kumar V.

A1 - Thompson,Andrew J.

A1 - Hothersall,J. Daniel

A1 - Connolly,Christopher N.

A1 - Lummis,Sarah C. R.

A1 - Lochner,Martin

AU - Simonin,Jonathan

AU - Vernekar,Sanjeev Kumar V.

AU - Thompson,Andrew J.

AU - Hothersall,J. Daniel

AU - Connolly,Christopher N.

AU - Lummis,Sarah C. R.

AU - Lochner,Martin

PY - 2012

Y1 - 2012

N2 - <p>The synthesis, photophysical and biological characterization of a small library of fluorescent 5-HT3 receptor ligands is described. Several of these novel granisetron conjugates have high quantum yields and show high affinity for the human 5-HT(3)AR. (C) 2011 Elsevier Ltd. All rights reserved.</p>

AB - <p>The synthesis, photophysical and biological characterization of a small library of fluorescent 5-HT3 receptor ligands is described. Several of these novel granisetron conjugates have high quantum yields and show high affinity for the human 5-HT(3)AR. (C) 2011 Elsevier Ltd. All rights reserved.</p>

KW - 5-HT3 receptor

KW - Cys-loop ligand-gated ion channels

KW - Fluorescent ligands

KW - Radioligand binding

KW - In vivo imaging

KW - ANTAGONISTS

KW - TARGET

U2 - 10.1016/j.bmcl.2011.11.097

DO - 10.1016/j.bmcl.2011.11.097

M1 - Article

JO - Bioorganic & Medicinal Chemistry Letters

JF - Bioorganic & Medicinal Chemistry Letters

SN - 0960-894X

IS - 2

VL - 22

SP - 1151

EP - 1155

ER -

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