Research output per year
Research output per year
Search results
-
2018
Impact of target warhead and linkage vector on inducing protein degradation: comparison of Bromodomain and Extra-Terminal (BET) degraders derived from triazolodiazepine (JQ1) and tetrahydroquinoline (I-BET726) BET inhibitor scaffolds
Chan, K. H., Zengerle, M., Testa, A. & Ciulli, A. (Lead / Corresponding author), 25 Jan 2018, In: Journal of Medicinal Chemistry. 61, 2, p. 504-513 10 p.Research output: Contribution to journal › Article › peer-review
Open AccessFile179 Citations (Scopus)396 Downloads (Pure) -
2017
Structural basis of PROTAC cooperative recognition for selective protein degradation
Gadd, M., Testa, A., Lucas, X., Chan, K. H., Chen, W., Lamont, D., Zengerle, M. & Ciulli, A. (Lead / Corresponding author), May 2017, In: Nature Chemical Biology. 13, 5, p. 514-521 11 p.Research output: Contribution to journal › Article › peer-review
Open AccessFile869 Citations (Scopus)723 Downloads (Pure) -
2016
Chemical genetics approaches for selective intervention in epigenetics
Runcie, A. C., Chan, K. H., Zengerle, M. & Ciulli, A. (Lead / Corresponding author), Aug 2016, In: Current Opinion in Chemical Biology. 33, p. 186-194 9 p.Research output: Contribution to journal › Review article › peer-review
Open AccessFile24 Citations (Scopus)284 Downloads (Pure)