Keyphrases
Targeted Protein Degradation
100%
E3 Ligase
100%
In Cis
66%
Ligase
66%
Proteolysis Targeting chimera (PROTAC)
66%
Bromodomain-containing Protein 4 (BRD4)
66%
DCAF16
33%
BRD4 Degradation
33%
Surface Complementarity
33%
Picomolar Potency
33%
Protein Domain
33%
E3 Ubiquitin Ligase
33%
Heterobifunctional Degrader
33%
Genetic Screening
33%
Proteasomal Degradation
33%
Ubiquitination
33%
Induced Proximity
33%
Structural Insights
33%
Molecular Glue
33%
Ubiquitin-mediated Degradation
33%
Degrader
33%
Reconstitution
33%
Conformational Change
33%
BRD2
33%
Bifunctional Compounds
33%
Mechanism of Action
33%
Rational Design
33%
Biophysical Characterization
33%
Biochemistry, Genetics and Molecular Biology
Ligase
100%
Protein Catabolism
100%
BRD4
60%
Ubiquitination
40%
Conformational Change
20%
Ubiquitin-Conjugating Enzyme
20%
BRD2
20%
Genetic Screening
20%
Protein Tertiary Structure
20%