Dissecting and Exploiting Molecular Recognition at Protein-Protein Interfaces (David Phillips Fellowship)

Project Details

StatusFinished
Effective start/end date8/04/137/07/15

Funding

  • Biotechnology and Biological Sciences Research Council (BB/G023123/2): £307,127.00

Research Output

Open Access
File
  • 30 Citations (Scopus)
    142 Downloads (Pure)

    Optimization of a “Bump-and-Hole” Approach to Allele-Selective BET Bromodomain Inhibition

    Runcie, A., Zengerle, M., Chan, K. H., Testa, A., Van Beurden, L., Baud, M., Epemolu, R., Ellis, L., Read, K., Coulthard, V., Brien, A. & Ciulli, A., 7 Mar 2018, In : Chemical Science. 9, 9, p. 2452-2468 17 p., 2452.

    Research output: Contribution to journalArticle

    Open Access
    File
  • 8 Citations (Scopus)
    166 Downloads (Pure)

    Allosteric targeting of the Fanconi anemia ubiquitin-conjugating enzyme Ube2T by fragment screening

    Morreale, F., Bortoluzzi, A., Chaugule, V., Arkinson, C., Walden, H. & Ciulli, A., 11 May 2017, In : Journal of Medicinal Chemistry. 60, 9, p. 4093-4098 6 p.

    Research output: Contribution to journalArticle

    Open Access
    File
  • 6 Citations (Scopus)
    164 Downloads (Pure)