European Lead Factory EUC2LID (IMI) (Joint with 29 other Partners)

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  • 2022

    IMI European Lead Factory - democratizing access to high-throughput screening

    Jones, P. S., Boucharens, S., McElroy, S. P., Morrison, A., Honarnejad, S., van Boeckel, S., van den Hurk, H., Basting, D., Hüser, J., Jaroch, S., Ottow, E., Benningshof, J., Folmer, R. H. A., Leemhuis, F., Kramer-Verhulst, P. M., Nies, V. J. M., Orrling, K. M., Rijnders, T., Pfander, C. & Engkvist, O. & 49 others, Pairaudeau, G., Simpson, P. B., Ortholand, J.-Y., Roche, D., Dömling, A., Kühnert, S. M., Roevens, P. W. M., van Vlijmen, H., van Wanrooij, E. J. A., Verbruggen, C., Nussbaumer, P., Ovaa, H., van der Stelt, M., Simonsen, K. B., Tagmose, L., Waldmann, H., Duffy, J., Finsinger, D., Jurzak, M., Burgess-Brown, N. A., Lee, W. H., Rutjes, F. P. J. T., Haag, H., Kallus, C., Mors, H., Dorval, T., Lesur, B., Ramon Olayo, F., Hamza, D., Jones, G., Pearce, C., Piechot, A., Tzalis, D., Clausen, M. H., Davis, J., Derouane, D., Vermeiren, C., Kaiser, M., Stockman, R. A., Barrault, D. V., Pannifer, A. D., Swedlow, J. R., Nelson, A. S., Orru, R. V. A., Ruijter, E., van Helden, S. P., Li, V. M., Vries, T. & de Vlieger, J. S. B., Apr 2022, In: Nature reviews. Drug discovery. 21, p. 245-246 2 p.

    Research output: Contribution to journalComment/debatepeer-review

    2 Citations (Scopus)
  • Imitation of β-lactam binding enables broad-spectrum metallo-β-lactamase inhibitors

    Brem, J. (Lead / Corresponding author), Panduwawala, T., Hansen, J. U., Hewitt, J., Liepins, E., Donets, P., Espina, L., Farley, A. J. M., Shubin, K., Campillos, G. G., Kiuru, P., Shishodia, S., Krahn, D., Leśniak, R. K., Schmidt (Adrian), J., Calvopiña, K., Turrientes, M.-C., Kavanagh, M. E., Lubriks, D. & Hinchliffe, P. & 41 others, Langley, G. W., Aboklaish, A. F., Eneroth, A., Backlund, M., Baran, A. G., Nielsen, E. I., Speake, M., Kuka, J., Robinson, J., Grinberga, S., Robinson, L., McDonough, M. A., Rydzik, A. M., Leissing, T. M., Jimenez-Castellanos, J. C., Avison, M. B., Da Silva Pinto, S., Pannifer, A. D., Martjuga, M., Widlake, E., Priede, M., Hopkins Navratilova, I., Gniadkowski, M., Belfrage, A. K., Brandt, P., Yli-Kauhaluoma, J., Bacque, E., Page, M. G. P., Björkling, F., Tyrrell, J. M., Spencer, J., Lang, P. A., Baranczewski, P., Cantón, R., McElroy, S. P., Jones, P. S., Baquero, F., Suna, E., Morrison, A., Walsh, T. R. & Schofield, C. J. (Lead / Corresponding author), Jan 2022, In: Nature Chemistry. 14, p. 15-24 10 p.

    Research output: Contribution to journalArticlepeer-review

    46 Citations (Scopus)