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• Synthesis of beta-D-Galp-(1 -> 4)-alpha-D-Manp methanephosphonate, a substrate analogue for the elongating alpha-D-mannosyl phosphate transferase in the Leishmania

  Borodkin, V. S., Ferguson, M. A. J. & Nikolaev, A. V., 30 Jul 2001, In: Tetrahedron Letters. 42, 31, p. 5305-5308 4 p.

  Research output: Contribution to journal › Article › peer-review
  16 Citations (Scopus)

• Synthesis of a Series of Diaminoindoles

  Martin, J. S., Mackenzie, C. J. & Gilbert, I. H., 3 Sep 2021, In: Journal of Organic Chemistry. 86, 17, p. 11333-11340 8 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

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  1 Citation (Scopus)

  42 Downloads (Pure)

• Synthesis of a partially protected 1D-6-O-(2-azido-2-deoxy-α-D-glucopyranosyl)-myo-inositol: a useful precursor of glycosylphosphatidylinositols and related compounds

  Cottaz, S., Brimacombe, J. S. & Ferguson, M. A. J., 1 Jan 1995, In: Carbohydrate Research. 270, 1, p. 85-91 7 p.

  Research output: Contribution to journal › Article › peer-review
  19 Citations (Scopus)

• Synthesis of an IGD peptidomimetic with motogenic activity

  Shpiro, N., Ellis, I. R., Dines, T. J., Schor, A. M., Schor, S. L., Norman, D. G. & Marquez, R., 2005, In: Molecular BioSystems. 1, 4, p. 318-320 3 p.

  Research output: Contribution to journal › Article › peer-review
  5 Citations (Scopus)

• Synthesis of an azido-tagged low affinity ratiometric calcium sensor

  Caldwell, S. T., Cairns, A. G., Olson, M., Chalmers, S., Sandison, M., Mullen, W., McCarron, J. G. & Hartley, R. C., 23 Dec 2015, In: Tetrahedron. 71, 51, p. 9571-9578 8 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File
  4 Citations (Scopus)

  30 Downloads (Pure)

• Synthesis of analogues of Congo red and evaluation of their anti-prion activity

  Sellarajah, S., Lekishvili, T., Bowring, C., Thompsett, A. R., Rudyk, H., Birkett, C. R., Brown, D. R. & Gilbert, I. H., 2004, In: Journal of Medicinal Chemistry. 47, 22, p. 5515-5534 20 p.

  Research output: Contribution to journal › Article › peer-review
  62 Citations (Scopus)

• Synthesis of aminoacids derivatives as Rev-RRE binding inhibitors, using solid phase combinatorial chemistry

  Jimenez-Bueno, G., Simons, C. & Gilbert, I. H., 2000.

  Research output: Contribution to conference › Poster

• Synthesis of aminoacids derivatives as Rev-RRE binding inhibitors, using solid phase combinatorial chemistry

  Jimenez-Bueno, G., Simons, C. & Gilbert, I. H., 2000, In: Antiviral Research. 46, 1, p. A43-A43 1 p., 26.

  Research output: Contribution to journal › Meeting abstract › peer-review

• Synthesis of allylamines in enantiomerically pure form

  Concellón, J. M., Baragaña, B. & Riego, E., 8 Jun 2000, In: Tetrahedron Letters. 41, 22, p. 4361-4362 2 p.

  Research output: Contribution to journal › Article › peer-review
  7 Citations (Scopus)

• Synthesis of a homochiral α,α-disubstituted α,β-diamino-acid

  Jolles, R. C. F., Crockett, A. K., Rees, D. C. & Gilbert, I., 1994, In: Tetrahedron: Asymmetry. 5, 9, p. 1661-1664 4 p.

  Research output: Contribution to journal › Comment/debate › peer-review
  21 Citations (Scopus)

• Synthesis of a cell-permeable analogue of a glycosylphosphatidylinositol (GPI) intermediate that is toxic to the living bloodstream form of Trypanosoma brucei

  Crossman, A., Smith, T. K., Ferguson, M. A. J. & Brimacombe, J. S., 24 Oct 2005, In: Tetrahedron Letters. 46, 43, p. 7419-7421 3 p.

  Research output: Contribution to journal › Article › peer-review
  6 Citations (Scopus)

• Synthesis of 6-N-biotinylaminohexyl isopropyl phosphorofluoridate: a potent tool for the inhibition/isolation of serine esterases and proteases

  Higson, A. P., Ferguson, M. A. J. & Nikolaev, A. V., Mar 1999, In: Synthesis-Stuttgart. 3, p. 407-409 3 p.

  Research output: Contribution to journal › Article › peer-review
  6 Citations (Scopus)

• Synthesis of 3-alkyl naphthalenes as novel estrogen receptor ligands

  Fang, J., Akwabi-Ameyaw, A., Britton, J. E., Katamreddy, S. R., Navas III, F., Miller, A. B., Williams, S. P., Gray, D. W., Orband-Miller, L. A., Shearin, J. & Heyer, D., 15 Sep 2008, In: Bioorganic & Medicinal Chemistry Letters. 18, 18, p. 5075-5077 3 p.

  Research output: Contribution to journal › Article › peer-review
  23 Citations (Scopus)

• Synthesis of 3 '-, 4 '- and 6 '-deoxy and other analogues of D-glucosaminylphosphatidylinositol

  Borissow, C. N., Smith, T. K., Ferguson, M. A. J. & Brimacombe, J. S., 1 Jan 2001, In: Tetrahedron Letters. 42, 1, p. 121-123 3 p.

  Research output: Contribution to journal › Article › peer-review
  5 Citations (Scopus)

• Synthesis of 3,3-disubstituted heterocycles by Pd-catalyzed arylallylation of unactivated alkenes

  Phillips, D., Hewitt, J. F. M. & France, D. J., 31 Jul 2018, In: ACS Omega. 3, 7, p. 8451-8459 9 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

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  4 Citations (Scopus)

  55 Downloads (Pure)

• Synthesis of 2-quinuclidonium by eliminating water: experimental quantification of the high basicity of extremely twisted amides

  Ly, T., Krout, M., Pham, D. K., Tani, K., Stoltz, B. M. & Julian, R. R., 21 Feb 2007, In: Journal of the American Chemical Society. 129, 7, p. 1864-1865 2 p.

  Research output: Contribution to journal › Article › peer-review
  30 Citations (Scopus)

• Synthesis of 1′-(4′-Thio-β-d-Ribofuranosyl) Uracil

  Guinan, M., Miller, G. J., Lynch, D. & Smith, M., 2021, Carbohydrate Chemistry: Proven Synthetic Methods. Kosma, P., Wrodnigg, T. & Stütz, A. (eds.). 1 ed. Boca Raton: CRC Press, Vol. 5. 6 p.

  Research output: Chapter in Book/Report/Conference proceeding › Chapter (peer-reviewed) › peer-review

• Synthesis of 1-D-6-O-[2-(N-hydroxyaminocarbonyl)amino-2-deoxy-alpha-D-glucopyranosyl]-myo-inositol 1-(n-octadecyl phosphate): a potential metalloenzyme inhibitor of glycosylphosphatidylinositol biosynthesis

  Crossman, A. T., Urbaniak, M. D. & Ferguson, M. A. J., 7 Jul 2008, In: Carbohydrate Research. 343, 9, p. 1478-1481 4 p.

  Research output: Contribution to journal › Article › peer-review
  7 Citations (Scopus)

• Synthesis of ¹³C₂¹⁵N₂-labeled anti-inflammatory and cytoprotective tricyclic bis(cyanoenone) ([¹³C₂¹⁵N₂]-TBE-31) as an internal standard for quantification by stable isotope dilution LC-MS method

  Zheng, S., Huang, J. T. -J., Knatko, E. V., Sharp, S., Higgins, M., Ojima, I., Dinkova-Kostova, A. T. & Honda, T., Aug 2014, In: Journal of Labelled Compounds and Radiopharmaceuticals. 57, 10, p. 606-610 5 p.

  Research output: Contribution to journal › Article › peer-review
  3 Citations (Scopus)

• Synthesis of (R)-2-methyl-4-deoxy and (R)-2-methyl-4,5-dideoxy analogues of 6-phosphogluconate as potential inhibitors of 6-phosphogluconate dehydrogenase

  Dardonville, C. & Gilbert, I. H., 2003, In: Organic and Biomolecular Chemistry. 1, 3, p. 552-559 8 p.

  Research output: Contribution to journal › Article › peer-review
  11 Citations (Scopus)

• Synthesis of (-)-(S, S)-clemastine by invertive N → C aryl migration in a lithiated carbamate

  Fournier, A. M., Brown, R. A., Farnaby, W., Miyatake-Ondozabal, H. & Clayden, J., 21 May 2010, In: Organic Letters. 12, 10, p. 2222-2225 4 p.

  Research output: Contribution to journal › Article › peer-review
  52 Citations (Scopus)

• Synthesising interconnections

  Fiadeiro, J. L., Lopes, A. & Maibaum, T. S. E., 1997, Algorithmic Languages and Calculi. Bird, R. S. & Meertens, L. (eds.). Springer , p. 240-264 25 p. (IFIP Advances in Information and Communication Technology).

  Research output: Chapter in Book/Report/Conference proceeding › Conference contribution

• Synthesis and use of the protein phosphatase affinity matrices microcystin-sepharose and microcystin-biotin-sepharose

  Moorhead, G. B. G., Haystead, T. A. J. & MacKintosh, C., 1 Dec 2007, Protein Phosphatase Protocols. Moorhead, G. (ed.). Springer , p. 39-45 7 p. (Methods in Molecular Biology; vol. 365).

  Research output: Chapter in Book/Report/Conference proceeding › Chapter
  9 Citations (Scopus)

• Synthesis and testing of peptides for anti-prion activity

  Sellarajah, S., Boussard, C., Lekishvili, T., Brown, D. R. & Gilbert, I. H., Nov 2008, In: European Journal of Medicinal Chemistry. 43, 11, p. 2418-2427 10 p.

  Research output: Contribution to journal › Article › peer-review
  3 Citations (Scopus)

• Synthesis and testing of 5-benzyl-2,4-diaminopyrimidines as potential inhibitors of leishmanial and trypanosomal dihydrofolate reductase

  Chowdhury, S. F., Hurtado Guerrero, R., Brun, R., Ruiz-Perez, L. M., Gonzalez Pacanowska, D. & Gilbert, I. H., 2002, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 17, 5, p. 293-302 10 p.

  Research output: Contribution to journal › Article › peer-review
  22 Citations (Scopus)

• Synthesis and structure-based dissection of cyclic peptide chitinase inhibitors: new leads for antifungal and anti-inflammatory drugs

  Dixon, M. J., Nathubhai, A., Andersen, O. A., van Aalten, D. M. F. & Eggleston, I. M., 2009, Peptides for youth: the proceedings of the 20th American Peptide Symposium. Del Valle, S., Escher, E. & Lubell, W. D. (eds.). New York: Springer , p. 525-526 2 p. (Advances in experimental medicine and biology; vol. 611).

  Research output: Chapter in Book/Report/Conference proceeding › Chapter
  2 Citations (Scopus)

• Synthesis and structure-activity relationships of a novel series of pyrimidines as potent inhibitors of TBK1/IKKε kinases

  McIver, E. G., Bryans, J., Birchall, K., Chugh, J., Drake, T., Lewis, S. J., Osborne, J., Smiljanic-Hurley, E., Tsang, W., Kamal, A., Levy, A., Newman, M., Taylor, D., Arthur, J. S. C., Clark, K. & Cohen, P., Dec 2012, In: Bioorganic & Medicinal Chemistry Letters. 22, 23, p. 7169-7173 5 p.

  Research output: Contribution to journal › Article › peer-review
  32 Citations (Scopus)

• Synthesis and preliminary assessment of the anticancer and Wnt/β-catenin inhibitory activity of small amide libraries of fenamates and profens

  Mathew, B., Hobrath, J. V., Lu, W., Li, Y. & Reynolds, R. C., Nov 2017, In: Medicinal Chemistry Research. 26, 11, p. 3038-3045 8 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

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  9 Citations (Scopus)

  161 Downloads (Pure)

• Synthesis and Optical Characterization of Anatase-TiO2 Nanowires by Hydrothermal Method

  Bakhshayesh, A., Dadar, H. & Mohammadi, M. R., Apr 2012, 4th International Conference on Nanostructures: (ICNS4). Iran

  Research output: Chapter in Book/Report/Conference proceeding › Conference contribution

• Synthesis and NAD(P)H: Quinone oxidoreductase 1 inducer activity of acetamide and pyridine-3-carbonitrile derivatives

  Ghorab, M. M., Shahat, A. A., Alsaid, M. S., Higgins, M., Dinkova-Kostova, A. T. & Naser, A. A., 2016, In: Biomedical Research. 27, 4, p. 1045-1048 4 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File
  49 Downloads (Pure)

• Synthesis and in vitro biochemical evaluation of oxime bond-linked daunorubicin-GnRH-III conjugates developed for targeted drug delivery

  Schuster, S., Biri-Kovács, B., Szeder, B., Farkas, V., Buday, L., Szabó, Z., Halmos, G. & Mező, G., 4 Apr 2018, In: Beilstein Journal of Organic Chemistry. 14, p. 756-771 16 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File
  15 Citations (Scopus)

  31 Downloads (Pure)

• Synthesis and inclusion study of a novel γ-cyclodextrin derivative as a potential thermo-sensitive carrier for doxorubicin

  Xu, D., Wang, L., Gourevich, D., Kabha, E., Arditti, F., Athamna, M., Cochran, S., Melzer, A. & Gnaim, J. M., Jul 2014, In: Chemical and Pharmaceutical Bulletin. 62, 7, p. 627-635 9 p.

  Research output: Contribution to journal › Article › peer-review
  6 Citations (Scopus)

• Synthesis and Evaluation of α-Thymidine Analogues as Novel Antimalarials

  Cui, H., Carrero-Lérida, J., Silva, A. P. G., Whittingham, J. L., Brannigan, J. A., Ruiz-Pérez, L. M., Read, K. D., Wilson, K. S., González-Pacanowska, D. & Gilbert, I. H., 2012, In: Journal of Medicinal Chemistry. 55, 24, p. 10948-57 10 p.

  Research output: Contribution to journal › Article › peer-review
  34 Citations (Scopus)

• Synthesis and Evaluation of Indatraline-Based Inhibitors for Trypanothione Reductase

  Walton, J. G. A., Jones, D. C., Kiuru, P., Durie, A. J., Westwood, N. J. & Fairlamb, A. H., 7 Feb 2011, In: ChemMedChem. 6, 2, p. 321-328 8 p.

  Research output: Contribution to journal › Article › peer-review
  22 Citations (Scopus)

• Synthesis and evaluation of analogues of congo red as potential compounds against transmissible spongiform. encephalopathies

  Rudyk, H., Knaggs, M. H., Vasiljevic, S., Hope, J., Birkett, C. & Gilbert, I. H., 2003, In: European Journal of Medicinal Chemistry. 38, 6, p. 567-579 13 p.

  Research output: Contribution to journal › Article › peer-review
  45 Citations (Scopus)

• Synthesis and evaluation of 9,9-dimethylxanthene tricyclics against trypanothione reductase, Trypanosoma brucei, Trypanosoma cruzi and Leishmania donovani

  Chibale, K., Visser, M., Yardley, V., Croft, S. L. & Fairlamb, A. H., 5 Jun 2000, In: Bioorganic and Medicinal Chemistry Letters. 10, 11, p. 1147-1150 4 p.

  Research output: Contribution to journal › Article › peer-review
  22 Citations (Scopus)

• Synthesis and Evaluation of 1-(1-(Benzo[b]thiophen-2-yl)cyclohexyl)piperidine (BTCP) Analogues as Inhibitors of Trypanothione Reductase

  Patterson, S., Jones, D. C., Shanks, E. J., Frearson, J. A., Gilbert, I. H., Wyatt, P. G. & Fairlamb, A. H., Aug 2009, In: ChemMedChem. 4, 8, p. 1341-1353 13 p.

  Research output: Contribution to journal › Article › peer-review
  50 Citations (Scopus)

• Synthesis and enzymology of modified N-benzyloxycarbonyl-L-cysteinylglycyl-3,3-dimethylaminopropylamide disulphides as alternative substrates for trypanothione reductase from Trypanosoma cruzi: Part 3

  Yuen, C. T., Garforth, J., Besheya, T., Jaouhari, R., McKie, J. H., Fairlamb, A. H. & Douglas, K. T., Jun 1999, In: Amino Acids. 17, 2, p. 175-183 9 p.

  Research output: Contribution to journal › Article › peer-review
  6 Citations (Scopus)

• Synthesis and crystallization of lead-zirconium-titanate (PZT) nanotubes at the low temperature using carbon nanotubes (CNTs) as sacrificial templates

  Mohammadi, M. R., Tabei, S. A., Nemati, A., Eder, D. & Pradeep, T., Sep 2012, In: Advanced Powder Technology. 23, 5, p. 647-654 8 p.

  Research output: Contribution to journal › Article › peer-review
  8 Citations (Scopus)

• Synthesis and characterization of quantum dots designed for biomedical use

  Kuzyniak, W., Adegoke, O., Sekhosana, K., D'Souza, S., Tshangana, S. C., Hoffmann, B., Ermilov, E. A., Nyokong, T. & Höpfner, M., 15 May 2014, In: International Journal of Pharmaceutics. 466, 1-2, p. 382-389 8 p.

  Research output: Contribution to journal › Article › peer-review
  30 Citations (Scopus)

• Synthesis and characterization of an iodinated bile-salt derivative for photoaffinity-labeling

  Henderson, C. J. & Percy-Robb, I. W., 12 Sep 1984, In: Biochimica et Biophysica Acta. Lipids and Lipid Metabolism. 795, 2, p. 257-264 8 p.

  Research output: Contribution to journal › Article › peer-review
  2 Citations (Scopus)

• Synthesis and characterisation of nanostructured neodymium titanium oxides by sol-gel process: Controlling the phase composition, crystal structure and grain size

  Mohammadi, M. R. & Fray, D. J., 1 Aug 2010, In: Materials Chemistry and Physics. 122, 2-3, p. 512-523 12 p.

  Research output: Contribution to journal › Article › peer-review
  14 Citations (Scopus)

• Synthesis and characterisation of nanosized TiO₂-ZrO₂ binary system prepared by an aqueous sol-gel process: Physical and sensing properties

  Mohammadi, M. R. & Fray, D. J., 20 Jul 2011, In: Sensors and Actuators, B: Chemical. 155, 2, p. 568-576 9 p.

  Research output: Contribution to journal › Article › peer-review
  39 Citations (Scopus)

• Synthesis and Characterisation of CNT-PZT Hybrid Material and PZT Nanotube by Sol-Gel Process

  Mohammadi, M. R. & Tabei, A., 12 Sep 2010, 7th International Conference on Inorganic Materials . Biarritz, France, p. P2.3 1 p.

  Research output: Chapter in Book/Report/Conference proceeding › Conference contribution

• Synthesis and biological properties of bioreductively targeted nitrothienyl prodrugs of combretastatin A-4

  Thomson, P., Naylor, M. A., Everett, S. A., Stratford, M. R. L., Lewis, G., Hill, S., Patel, K. B., Wardman, P. & Davis, P. D., Nov 2006, In: Molecular Cancer Therapeutics. 5, 11, p. 2886-2894 9 p.

  Research output: Contribution to journal › Article › peer-review
  36 Citations (Scopus)

• Synthesis and Biological Investigation of (+)-JD1, an Organometallic BET Bromodomain Inhibitor

  Hassell-Hart, S., Runcie, A., Krojer, T., Doyle, J., Lineham, E., Ocasio, C. A., Neto, B. A. D., Fedorov, O., Marsh, G., Maple, H., Felix, R., Banks, R., Ciulli, A., Picaud, S., Filippakopoulos, P., Von Delft, F., Brennan, P., Stewart, H. J. S., Chevassut, T. J., Walker, M., & 3 othersAustin, C., Morley, S. & Spencer, J., 10 Feb 2020, In: Organometallics. 39, 3

  Research output: Contribution to journal › Article › peer-review
  4 Citations (Scopus)

• Synthesis and biological evaluation of phosphate Prodrugs of 4-Phospho-D-erythronohydroxamic acid, an inhibitor of 6-phosphogluconate dehydrogenase

  Ruda, G. F., Alibu, V. P., Mitsos, C., Bidet, O., Kaiser, M., Brun, R., Barrett, M. P. & Gilbert, I. H., Aug 2007, In: ChemMedChem. 2, 8, p. 1169-1180 12 p.

  Research output: Contribution to journal › Article › peer-review
  26 Citations (Scopus)

  9 Downloads (Pure)

• Synthesis and biological evaluation of novel 2-phenylquinazoline-4-amine derivatives: identification of 6-phenyl-8H-benzo[g]quinazolino[4,3-b]quinazolin-8-one as a highly potent inducer of NAD(P)H quinone oxidoreductase 1

  Ghorab, M. M., Alsaid, M. S., El-Gazzar, M. G., Higgins, M., Dinkova-Kostova, A. T. & Shahat, A. A., 2016, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 31, Suppl. 1, p. 34-49 6 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File
  4 Citations (Scopus)

  205 Downloads (Pure)

• Synthesis and biological evaluation of biotin conjugates of (±)-(4bS,8aR,10aS)-10a-ethynyl-4b,8,8-trimethyl-3,7-dioxo-3,4b,7,8,8a,9,10,10a-octahydro-phenanthrene-2,6-dicarbonitrile, an activator of the Keap1/Nrf2/ARE pathway, for the isolation of its protein targets

  Saito, A., Higgins, M., Zheng, S., Li, W., Ojima, I., Dinkova-Kostova, A. T. & Honda, T., 15 Oct 2013, In: Bioorganic & Medicinal Chemistry Letters. 23, 20, p. 5540-5543 4 p.

  Research output: Contribution to journal › Article › peer-review
  5 Citations (Scopus)

• Synthesis and biological evaluation of 1-[2-cyano-3,12-dioxooleana-1,9(11)-dien-28-oyl]-4-ethynylimidazole. A novel and highly potent anti-inflammatory and cytoprotective agent

  Honda, T., Dinkova-Kostova, A. T., David, E., Padegimas, E. M., Sundararajan, C., Visnick, M., Bumeister, R. & Wigley, W. C., 15 Apr 2011, In: Bioorganic & Medicinal Chemistry Letters. 21, 8, p. 2188-2191 4 p.

  Research output: Contribution to journal › Article › peer-review
  20 Citations (Scopus)