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  Synthesis and inclusion study of a novel γ-cyclodextrin derivative as a potential thermo-sensitive carrier for doxorubicin

  Xu, D., Wang, L., Gourevich, D., Kabha, E., Arditti, F., Athamna, M., Cochran, S., Melzer, A. & Gnaim, J. M., Jul 2014, In: Chemical and Pharmaceutical Bulletin. 62, 7, p. 627-635 9 p.

  Research output: Contribution to journal › Article › peer-review
  6 Citations (Scopus)

• Synthesis and in vitro biochemical evaluation of oxime bond-linked daunorubicin-GnRH-III conjugates developed for targeted drug delivery

  Schuster, S., Biri-Kovács, B., Szeder, B., Farkas, V., Buday, L., Szabó, Z., Halmos, G. & Mező, G., 4 Apr 2018, In: Beilstein Journal of Organic Chemistry. 14, p. 756-771 16 p.

  Research output: Contribution to journal › Article › peer-review

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  17 Citations (Scopus)

  35 Downloads (Pure)

• Synthesis and NAD(P)H: Quinone oxidoreductase 1 inducer activity of acetamide and pyridine-3-carbonitrile derivatives

  Ghorab, M. M., Shahat, A. A., Alsaid, M. S., Higgins, M., Dinkova-Kostova, A. T. & Naser, A. A., 2016, In: Biomedical Research. 27, 4, p. 1045-1048 4 p.

  Research output: Contribution to journal › Article › peer-review

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• Synthesis and preliminary assessment of the anticancer and Wnt/β-catenin inhibitory activity of small amide libraries of fenamates and profens

  Mathew, B., Hobrath, J. V., Lu, W., Li, Y. & Reynolds, R. C., Nov 2017, In: Medicinal Chemistry Research. 26, 11, p. 3038-3045 8 p.

  Research output: Contribution to journal › Article › peer-review

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  10 Citations (Scopus)

  166 Downloads (Pure)

• Synthesis and structure-activity relationships of a novel series of pyrimidines as potent inhibitors of TBK1/IKKε kinases

  McIver, E. G., Bryans, J., Birchall, K., Chugh, J., Drake, T., Lewis, S. J., Osborne, J., Smiljanic-Hurley, E., Tsang, W., Kamal, A., Levy, A., Newman, M., Taylor, D., Arthur, J. S. C., Clark, K. & Cohen, P., Dec 2012, In: Bioorganic & Medicinal Chemistry Letters. 22, 23, p. 7169-7173 5 p.

  Research output: Contribution to journal › Article › peer-review
  32 Citations (Scopus)

• Synthesis and testing of 5-benzyl-2,4-diaminopyrimidines as potential inhibitors of leishmanial and trypanosomal dihydrofolate reductase

  Chowdhury, S. F., Hurtado Guerrero, R., Brun, R., Ruiz-Perez, L. M., Gonzalez Pacanowska, D. & Gilbert, I. H., 2002, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 17, 5, p. 293-302 10 p.

  Research output: Contribution to journal › Article › peer-review
  17 Citations (Scopus)

• Synthesis and testing of peptides for anti-prion activity

  Sellarajah, S., Boussard, C., Lekishvili, T., Brown, D. R. & Gilbert, I. H., Nov 2008, In: European Journal of Medicinal Chemistry. 43, 11, p. 2418-2427 10 p.

  Research output: Contribution to journal › Article › peer-review
  3 Citations (Scopus)

• Synthesis of (-)-(S, S)-clemastine by invertive N → C aryl migration in a lithiated carbamate

  Fournier, A. M., Brown, R. A., Farnaby, W., Miyatake-Ondozabal, H. & Clayden, J., 21 May 2010, In: Organic Letters. 12, 10, p. 2222-2225 4 p.

  Research output: Contribution to journal › Article › peer-review
  52 Citations (Scopus)

• Synthesis of (R)-2-methyl-4-deoxy and (R)-2-methyl-4,5-dideoxy analogues of 6-phosphogluconate as potential inhibitors of 6-phosphogluconate dehydrogenase

  Dardonville, C. & Gilbert, I. H., 2003, In: Organic and Biomolecular Chemistry. 1, 3, p. 552-559 8 p.

  Research output: Contribution to journal › Article › peer-review
  6 Citations (Scopus)

• Synthesis of ¹³C₂¹⁵N₂-labeled anti-inflammatory and cytoprotective tricyclic bis(cyanoenone) ([¹³C₂¹⁵N₂]-TBE-31) as an internal standard for quantification by stable isotope dilution LC-MS method

  Zheng, S., Huang, J. T. -J., Knatko, E. V., Sharp, S., Higgins, M., Ojima, I., Dinkova-Kostova, A. T. & Honda, T., Aug 2014, In: Journal of Labelled Compounds and Radiopharmaceuticals. 57, 10, p. 606-610 5 p.

  Research output: Contribution to journal › Article › peer-review
  3 Citations (Scopus)

• Synthesis of 1-D-6-O-[2-(N-hydroxyaminocarbonyl)amino-2-deoxy-alpha-D-glucopyranosyl]-myo-inositol 1-(n-octadecyl phosphate): a potential metalloenzyme inhibitor of glycosylphosphatidylinositol biosynthesis

  Crossman, A. T., Urbaniak, M. D. & Ferguson, M. A. J., 7 Jul 2008, In: Carbohydrate Research. 343, 9, p. 1478-1481 4 p.

  Research output: Contribution to journal › Article › peer-review
  7 Citations (Scopus)

• Synthesis of 2-quinuclidonium by eliminating water: experimental quantification of the high basicity of extremely twisted amides

  Ly, T., Krout, M., Pham, D. K., Tani, K., Stoltz, B. M. & Julian, R. R., 21 Feb 2007, In: Journal of the American Chemical Society. 129, 7, p. 1864-1865 2 p.

  Research output: Contribution to journal › Article › peer-review
  31 Citations (Scopus)

• Synthesis of 3,3-disubstituted heterocycles by Pd-catalyzed arylallylation of unactivated alkenes

  Phillips, D., Hewitt, J. F. M. & France, D. J., 31 Jul 2018, In: ACS Omega. 3, 7, p. 8451-8459 9 p.

  Research output: Contribution to journal › Article › peer-review

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  4 Citations (Scopus)

  57 Downloads (Pure)

• Synthesis of 3 '-, 4 '- and 6 '-deoxy and other analogues of D-glucosaminylphosphatidylinositol

  Borissow, C. N., Smith, T. K., Ferguson, M. A. J. & Brimacombe, J. S., 1 Jan 2001, In: Tetrahedron Letters. 42, 1, p. 121-123 3 p.

  Research output: Contribution to journal › Article › peer-review
  5 Citations (Scopus)

• Synthesis of 3-alkyl naphthalenes as novel estrogen receptor ligands

  Fang, J., Akwabi-Ameyaw, A., Britton, J. E., Katamreddy, S. R., Navas III, F., Miller, A. B., Williams, S. P., Gray, D. W., Orband-Miller, L. A., Shearin, J. & Heyer, D., 15 Sept 2008, In: Bioorganic & Medicinal Chemistry Letters. 18, 18, p. 5075-5077 3 p.

  Research output: Contribution to journal › Article › peer-review
  24 Citations (Scopus)

• Synthesis of 6-N-biotinylaminohexyl isopropyl phosphorofluoridate: a potent tool for the inhibition/isolation of serine esterases and proteases

  Higson, A. P., Ferguson, M. A. J. & Nikolaev, A. V., Mar 1999, In: Synthesis-Stuttgart. 3, p. 407-409 3 p.

  Research output: Contribution to journal › Article › peer-review
  5 Citations (Scopus)

• Synthesis of a cell-permeable analogue of a glycosylphosphatidylinositol (GPI) intermediate that is toxic to the living bloodstream form of Trypanosoma brucei

  Crossman, A., Smith, T. K., Ferguson, M. A. J. & Brimacombe, J. S., 24 Oct 2005, In: Tetrahedron Letters. 46, 43, p. 7419-7421 3 p.

  Research output: Contribution to journal › Article › peer-review
  6 Citations (Scopus)

• Synthesis of allylamines in enantiomerically pure form

  Concellón, J. M., Baragaña, B. & Riego, E., 8 Jun 2000, In: Tetrahedron Letters. 41, 22, p. 4361-4362 2 p.

  Research output: Contribution to journal › Article › peer-review
  1 Citation (Scopus)

• Synthesis of analogues of Congo red and evaluation of their anti-prion activity

  Sellarajah, S., Lekishvili, T., Bowring, C., Thompsett, A. R., Rudyk, H., Birkett, C. R., Brown, D. R. & Gilbert, I. H., 2004, In: Journal of Medicinal Chemistry. 47, 22, p. 5515-5534 20 p.

  Research output: Contribution to journal › Article › peer-review
  62 Citations (Scopus)

• Synthesis of an azido-tagged low affinity ratiometric calcium sensor

  Caldwell, S. T., Cairns, A. G., Olson, M., Chalmers, S., Sandison, M., Mullen, W., McCarron, J. G. & Hartley, R. C., 23 Dec 2015, In: Tetrahedron. 71, 51, p. 9571-9578 8 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

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  4 Citations (Scopus)

  33 Downloads (Pure)

• Synthesis of an IGD peptidomimetic with motogenic activity

  Shpiro, N., Ellis, I. R., Dines, T. J., Schor, A. M., Schor, S. L., Norman, D. G. & Marquez, R., 2005, In: Molecular BioSystems. 1, 4, p. 318-320 3 p.

  Research output: Contribution to journal › Article › peer-review
  5 Citations (Scopus)

• Synthesis of a partially protected 1D-6-O-(2-azido-2-deoxy-α-D-glucopyranosyl)-myo-inositol: a useful precursor of glycosylphosphatidylinositols and related compounds

  Cottaz, S., Brimacombe, J. S. & Ferguson, M. A. J., 1 Jan 1995, In: Carbohydrate Research. 270, 1, p. 85-91 7 p.

  Research output: Contribution to journal › Article › peer-review
  19 Citations (Scopus)

• Synthesis of a Series of Diaminoindoles

  Martin, J. S., Mackenzie, C. J. & Gilbert, I. H., 3 Sept 2021, In: Journal of Organic Chemistry. 86, 17, p. 11333-11340 8 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

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  1 Citation (Scopus)

  52 Downloads (Pure)

• Synthesis of beta-D-Galp-(1 -> 4)-alpha-D-Manp methanephosphonate, a substrate analogue for the elongating alpha-D-mannosyl phosphate transferase in the Leishmania

  Borodkin, V. S., Ferguson, M. A. J. & Nikolaev, A. V., 30 Jul 2001, In: Tetrahedron Letters. 42, 31, p. 5305-5308 4 p.

  Research output: Contribution to journal › Article › peer-review
  16 Citations (Scopus)

• Synthesis of carbohydrate capped silicon nanoparticles and their reduced cytotoxicity, in vivo toxicity, and cellular uptake

  Ahire, J. H., Behray, M., Webster, C. A., Wang, Q., Sherwood, V., Saengkrit, N., Ruktanonchai, U., Woramongkolchai, N. & Chao, Y., 26 Aug 2015, In: Advanced Healthcare Materials. 4, 12, p. 1877-1886 10 p.

  Research output: Contribution to journal › Article › peer-review
  25 Citations (Scopus)

• Synthesis of Densely Functionalized N-Alkenyl 2-Pyridones via Benzyne-Induced Ring Opening of Thiazolino-Fused 2-Pyridones

  Singh, P., Cairns, A. G., Adolfsson, D. E., Ådén, J., Sauer, U. H. & Almqvist, F., 16 Sept 2019, In: Organic Letters. 21, 17, p. 6946-6950 5 p.

  Research output: Contribution to journal › Article › peer-review
  12 Citations (Scopus)

• Synthesis of enantiopure α'-amino α,β-epoxy ketones from α'-amino bromomethyl ketones

  Barluenga, J., Baragana, B., Concellón, J. M., Piñera-Nicolás, A., Rosario Díaz, M. & García-Granda, S., 9 Jul 1999, In: Journal of Organic Chemistry. 64, 14, p. 5048-5052 5 p.

  Research output: Contribution to journal › Article › peer-review
  12 Citations (Scopus)

• Synthesis of glycosaminoglycans by cloned bovine endothelial cells cultured on collagen gels

  Winterbourne, D. J., Schor, A. M. & Gallagher, J. T., Sept 1983, In: European Journal of Biochemistry. 135, 2, p. 271-7 7 p.

  Research output: Contribution to journal › Article › peer-review

• Synthesis of highly pure nanocrystalline and mesoporous CaTiO₃ by a particulate sol-gel route at the low temperature

  Mohammadi, M. R. & Fray, D. J., 18 Oct 2013, In: Journal of Sol-Gel Science and Technology. 68, 2, p. 324-333 10 p.

  Research output: Contribution to journal › Article › peer-review
  17 Citations (Scopus)

• Synthesis of high surface area nanocrystalline anatase-TiO₂ powders derived from particulate sol-gel route by tailoring processing parameters

  Mohammadi, M. R., Cordero-Cabrera, M. C., Ghorbani, M. & Fray, D. J., 1 Oct 2006, In: Journal of Sol-Gel Science and Technology. 40, 1, p. 15-23 9 p.

  Research output: Contribution to journal › Article › peer-review
  68 Citations (Scopus)

• Synthesis of Imidazole C1- and C3-Ribonucleoside Phosphoramidites for Probing Catalytic Mechanism in Ribozyme

  Harusawa, S., Fujii, K., Nishiura, M., Araki, L., Usami, Y., Zhao, Z. & Lilley, D. M. J., 1 Sept 2011, In: Heterocycles. 83, 9, p. 2041-2055 15 p.

  Research output: Contribution to journal › Article › peer-review
  9 Citations (Scopus)

• Synthesis of isomeric phosphoubiquitin chains reveals that phosphorylation controls deubiquitinase activity and specificity

  Huguenin-Dezot, N., De Cesare, V., Peltier, J., Knebel, A., Kristariyanto, Y. A., Rogerson, D. T., Kulathu, Y., Trost, M. & Chin, J. W., 26 Jul 2016, In: Cell Reports. 16, 4, p. 1180-1193 14 p.

  Research output: Contribution to journal › Article › peer-review

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  47 Citations (Scopus)

  156 Downloads (Pure)

• Synthesis of N-(4-chlorophenyl) substituted pyrano[2,3-c]pyrazoles enabling PKBβ/AKT2 inhibitory and in vitro anti-glioma activity

  Vala, R. M., Tandon, V., Nicely, L., Guo, L., Gu, Y., Banerjee, S. & Patel, H. M., 2022, In: Annals of Medicine. 54, 1, p. 2549-2561 13 p.

  Research output: Contribution to journal › Article › peer-review

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  3 Citations (Scopus)

  16 Downloads (Pure)

• Synthesis of nanostructured and nanoporous TiO₂-AgO mixed oxide derived from a particulate sol-gel route: Physical and sensing characteristics

  Mohammadi, M. R. & Fray, D. J., 1 Aug 2011, In: Metallurgical and Materials Transactions A. 42, 8, p. 2481-2492 12 p.

  Research output: Contribution to journal › Article › peer-review
  7 Citations (Scopus)

• Synthesis of nano β‐TCP and the effects on the mechanical and biological properties of β‐TCP/HDPE/UHMWPE nanocomposites

  Bagheri Hossein Abadi, M., Ghasemi, I., Khavandi, A., Shokrgozar, M. A., Farokhi, M., Homaeigohar, S. & Eslamifar, A., Oct 2010, In: Polymer composites. 31, 10, p. 1745-1753 9 p.

  Research output: Contribution to journal › Article › peer-review
  19 Citations (Scopus)

• Synthesis of N-benzyloxycarbonyl-l-cysteinylglycine 3-dimethylaminopropylamide disulfide: A cheap and convenient new assay for trypanothione reductase

  El-Waer, A., Douglas, K. T., Smith, K. & Fairlamb, A. H., Oct 1991, In: Analytical Biochemistry. 198, 1, p. 212-216 5 p.

  Research output: Contribution to journal › Article › peer-review
  18 Citations (Scopus)

• Synthesis of new shogaol analogues as NRF2 activators and evaluation of their anti-inflammatory activity, modes of action and metabolic stability

  Mak, K-K., Shiming, Z., Sakirolla, R., Balijepalli, M. K., Dinkova-Kostova, A. T., Epemolu, O., Mohd, Z. & Pichika, M. R., 13 Feb 2023, In: Antioxidants . 12, 2, 27 p., 475.

  Research output: Contribution to journal › Article › peer-review

  Open Access

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• Synthesis of Novel C4-Linked C-2-Imidazole Ribonucleoside Phosphoramidite and Its Application to Probing the Catalytic Mechanism of a Ribozyme

  Araki, L., Morita, K., Yamaguchi, M., Zhao, Z-Y., Wilson, T. J., Lilley, D. M. J. & Harusawa, S., 20 Mar 2009, In: Journal of Organic Chemistry. 74, 6, p. 2350-2356 7 p.

  Research output: Contribution to journal › Article › peer-review
  24 Citations (Scopus)

• Synthesis of novel glycosyl phosphate analogues: derivatives of an acceptor substrate for the Leishmania elongating alpha-D-mannopyranosylphosphate transferase

  Ross, A. J., Higson, A. P., Ferguson, M. A. J. & Nikolaev, A. V., 3 Sept 1999, In: Tetrahedron Letters. 40, 36, p. 6695-6698 4 p.

  Research output: Contribution to journal › Article › peer-review
  7 Citations (Scopus)

• Synthesis of novel tetrazole C5-linked C0- and C2-ribonucleoside phosphoramidites using MePOM and POM groups for probing RNA catalysis

  Harusawa, S., Yoneyama, H., Fujisue, D., Nishiura, M., Fujitake, M., Usami, Y., Zhao, Z., Mcphee, S. A., Wilson, T. J. & Lilley, D. M. J., 2012, In: Tetrahedron Letters. 53, 44, p. 5891-5894 4 p.

  Research output: Contribution to journal › Article › peer-review
  17 Citations (Scopus)

• Synthesis of oligomeric phosphono analogues of Leishmania lipophosphoglycan fragments

  Borodkin, V. S., Milne, F. C., Ferguson, M. A. J. & Nikolaev, A. V., 21 Oct 2002, In: Tetrahedron Letters. 43, 43, p. 7821-7825 5 p.

  Research output: Contribution to journal › Article › peer-review
  14 Citations (Scopus)

• Synthesis of potential bisubstrate inhibitors of Leishmania elongating α-d-mannosyl phosphate transferase

  Borodkin, V. S., Ferguson, M. A. J. & Nikolaev, A. V., 2004, In: Tetrahedron Letters. 45, 4, p. 857-862 6 p.

  Research output: Contribution to journal › Article › peer-review
  16 Citations (Scopus)

• Synthesis of potential metal-binding group compounds to examine the zinc dependency of the GPI de-N-acetylase metalloenzyme in Trypanosoma brucei

  Abdelwahab, N. Z., Urbaniak, M. D., Ferguson, M. A. J. & Crossman, A. T., 1 May 2011, In: Carbohydrate Research. 346, 6, p. 708-714 7 p.

  Research output: Contribution to journal › Article › peer-review
  6 Citations (Scopus)

• Synthesis of protected myo-inositols

  Gilbert, I. H., Holmes, A. B. & Young, R. C., 1990, In: Tetrahedron Letters. 31, 18, p. 2633-2634 2 p.

  Research output: Contribution to journal › Article › peer-review
  14 Citations (Scopus)

• Synthesis of some second-generation substrate analogues of early intermediates in the biosynthetic pathway of glycosylphosphatidylinositol membrane anchors

  Crossman Jr., A., Brimacombe, J. S., Ferguson, M. A. J. & Smith, T. K., 15 Sept 1999, In: Carbohydrate Research. 321, 1-2, p. 42-51 10 p.

  Research output: Contribution to journal › Article › peer-review
  18 Citations (Scopus)

• Synthesis of water-soluble sugar derivatives of combretastatin A-4

  Brown, R. T., Fox, B. W., Hadfield, J. A., McGown, A. T., Mayalarp, S. P., Pettit, G. R. & Woods, J. A., 1995, In: Journal of the Chemical Society - Perkin Transactions 1. 5, p. 577-581 5 p.

  Research output: Contribution to journal › Article › peer-review
  30 Citations (Scopus)

• Synthesis of Well-Defined, Surfactant-Free Co₃O₄ Nanoparticles: The Impact of Size and Manganese Promotion on Co₃O₄ Reduction and Water Oxidation Activity

  Pritchard, J., Morris, L., Walsh, D., Sadasivan, S., Ménard, H., Bellabarba, R. M., Weller, M. T. & Tooze, R. P., Jan 2018, In: Catalysis Letters. 148, 1, p. 235-245 11 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

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  4 Citations (Scopus)

  311 Downloads (Pure)

• Synthesis of β-keto and α,β-unsaturated N-acetylcysteamine thioesters

  Gilbert, I. H., Ginty, M., O'Neill, J. A., Simpson, T. J., Staunton, J. & Willis, C. L., 1995, In: Bioorganic & Medicinal Chemistry Letters. 5, 15, p. 1587-1590 4 p.

  Research output: Contribution to journal › Article › peer-review
  29 Citations (Scopus)

• Synthesizing efficacious genistein in conjugation with superparamagnetic Fe₃O₄ decorated with bio-compatible carboxymethylated chitosan against acute leukemia lymphoma

  Ghasemi Goorbandi, R., Mohammadi, M. R. & Malekzadeh, K., 20 Mar 2020, In: Biomaterials Research. 24, p. 1-13 13 p., 9.

  Research output: Contribution to journal › Article › peer-review

  Open Access

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  14 Citations (Scopus)

  65 Downloads (Pure)

• Synthetic anisomycin analogues activating the JNK/SAPK1 and p38/SAPK2 pathways

  Rosser, E. M., Morton, S., Ashton, K. S., Cohen, P. & Hulme, A. N., 7 Jan 2004, In: Organic and Biomolecular Chemistry. 2, 1, p. 142-149 8 p.

  Research output: Contribution to journal › Article › peer-review
  25 Citations (Scopus)