A bump-and-hole approach to engineer controlled selectivity of BET bromodomain chemical probes

Matthias G. J. Baud, Enrique Lin-Shiao, Teresa Cardote, Cynthia Tallant, Annica Pschibul, Kwok-Ho Chan, Michael Zengerle, Jordi R. Garcia, Terence T.-L. Kwan, Fleur M. Ferguson, Alessio Ciulli (Lead / Corresponding author)

    Research output: Contribution to journal › Article › peer-review

    121 Citations (Scopus)

    Fingerprint

    Dive into the research topics of 'A bump-and-hole approach to engineer controlled selectivity of BET bromodomain chemical probes'. Together they form a unique fingerprint.

    Keyphrases

    Pharmacology, Toxicology and Pharmaceutical Science

    Biochemistry, Genetics and Molecular Biology