A series of 4- and 6-substituted derivatives of benzyl N-acetyl-ß-D- glucosaminide were prepared and assessed as inhibitors of bovine ß-1,4- galactosyl transferase. Of the azido, amino, and acetamido compounds tested, only the 4-amino compound (2) produced significant inhibition of this enzyme.
Field, R. A., Neville, D. C. A., Smith, R. W., & Ferguson, M. A. J. (1994). Acceptor analogues as potential inhibitors of bovine β-1,4-galactosyl transferase. Bioorganic & Medicinal Chemistry Letters, 4(3), 391-394. https://doi.org/10.1016/0960-894X(94)80002-2