Anti-malarial agents

Ian Gilbert (Inventor), Neil Norcross (Inventor), Beatriz Baragana (Inventor), Achim Porzelle (Inventor)

    Research output: Patent

    Abstract

    The present invention relates to a novel class of quinolone-4-carboxamide Pf3D7 inhibitors of general formula (I) (Formula (I)) wherein R1, R2, R3, R4, R5, R6, R7, R8 and X are as defined herein, to their use in medicine, and in the treatment of malaria in particular, to compositions containing them, to processes for their preparation and to intermediates used in such processes.
    Original languageEnglish
    Patent numberPCT/GB2013/050633
    IPCC07D 215/52 (2006.01), A61K 31/4725 (2006.01), A61P 33/06 (2006.01)
    Publication statusPublished - 17 Oct 2013

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    4-Quinolones
    Antimalarials
    Patents and inventions
    Medicine
    Chemical analysis

    Cite this

    Gilbert, I., Norcross, N., Baragana, B., & Porzelle, A. (2013). IPC No. C07D 215/52 (2006.01), A61K 31/4725 (2006.01), A61P 33/06 (2006.01) . Anti-malarial agents. (Patent No. PCT/GB2013/050633).
    Gilbert, Ian (Inventor) ; Norcross, Neil (Inventor) ; Baragana, Beatriz (Inventor) ; Porzelle, Achim (Inventor). / Anti-malarial agents. IPC No.: C07D 215/52 (2006.01), A61K 31/4725 (2006.01), A61P 33/06 (2006.01) . Patent No.: PCT/GB2013/050633.
    @misc{5faeb126911a494abd794bf429d7fb7d,
    title = "Anti-malarial agents",
    abstract = "The present invention relates to a novel class of quinolone-4-carboxamide Pf3D7 inhibitors of general formula (I) (Formula (I)) wherein R1, R2, R3, R4, R5, R6, R7, R8 and X are as defined herein, to their use in medicine, and in the treatment of malaria in particular, to compositions containing them, to processes for their preparation and to intermediates used in such processes.",
    author = "Ian Gilbert and Neil Norcross and Beatriz Baragana and Achim Porzelle",
    year = "2013",
    month = "10",
    day = "17",
    language = "English",
    type = "Patent",
    note = "PCT/GB2013/050633; C07D 215/52 (2006.01), A61K 31/4725 (2006.01), A61P 33/06 (2006.01)",

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    Gilbert, I, Norcross, N, Baragana, B & Porzelle, A 2013, Anti-malarial agents, Patent No. PCT/GB2013/050633, IPC No. C07D 215/52 (2006.01), A61K 31/4725 (2006.01), A61P 33/06 (2006.01) .

    Anti-malarial agents. / Gilbert, Ian (Inventor); Norcross, Neil (Inventor); Baragana, Beatriz (Inventor); Porzelle, Achim (Inventor).

    IPC No.: C07D 215/52 (2006.01), A61K 31/4725 (2006.01), A61P 33/06 (2006.01) . Patent No.: PCT/GB2013/050633.

    Research output: Patent

    TY - PAT

    T1 - Anti-malarial agents

    AU - Gilbert, Ian

    AU - Norcross, Neil

    AU - Baragana, Beatriz

    AU - Porzelle, Achim

    PY - 2013/10/17

    Y1 - 2013/10/17

    N2 - The present invention relates to a novel class of quinolone-4-carboxamide Pf3D7 inhibitors of general formula (I) (Formula (I)) wherein R1, R2, R3, R4, R5, R6, R7, R8 and X are as defined herein, to their use in medicine, and in the treatment of malaria in particular, to compositions containing them, to processes for their preparation and to intermediates used in such processes.

    AB - The present invention relates to a novel class of quinolone-4-carboxamide Pf3D7 inhibitors of general formula (I) (Formula (I)) wherein R1, R2, R3, R4, R5, R6, R7, R8 and X are as defined herein, to their use in medicine, and in the treatment of malaria in particular, to compositions containing them, to processes for their preparation and to intermediates used in such processes.

    M3 - Patent

    M1 - PCT/GB2013/050633

    ER -

    Gilbert I, Norcross N, Baragana B, Porzelle A, inventors. Anti-malarial agents. C07D 215/52 (2006.01), A61K 31/4725 (2006.01), A61P 33/06 (2006.01) . 2013 Oct 17.