Optimization of a “Bump-and-Hole” Approach to Allele-Selective BET Bromodomain Inhibition

Andrew Runcie, Michael Zengerle, Kwok Ho Chan, Andrea Testa, Lars Van Beurden, Matthias Baud, Rafiu Epemolu, Lucy Ellis, Kevin Read, V. Coulthard, A. Brien, Alessio Ciulli (Lead / Corresponding author)

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34 Citations (Scopus)
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Keyphrases

Biochemistry, Genetics and Molecular Biology