Abstract
A method of selectively inhibiting a bromodomain in the presence of other bromodomains comprising introducing a functionally silent mutation into the bromodomain in the presence of other wild type bromodomains and selectively inhibiting the mutated bromodomain.
| Translated title of the contribution | Enzymes functional probes |
|---|---|
| Original language | French |
| Patent number | WO/2015/079259 |
| Priority date | 28/11/13 |
| Filing date | 28/11/14 |
| Publication status | Published - 4 Jun 2015 |