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Stereochemical inversion at a 1,4-cyclohexyl PROTAC linker fine-tunes conformation and binding affinity
Martina Pierri
, Xingui Liu
,
Alena Kroupova
,
Zoe Rutter
,
Alex J. Hallatt
,
Alessio Ciulli
(Lead / Corresponding author)
Centre for Targeted Protein Degradation
Biological Chemistry and Drug Discovery
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5
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157
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