The efflux pump ABCC1/MRP1 constitutively restricts PROTAC sensitivity in cancer cells

Gernot Wolf, Conner Craigon, Shao Thing Teoh, Patrick Essletzbichler, Svenja Onstein, Diane Cassidy, Esther C.H. Uijttewaal, Vojtech Dvorak, Yuting Cao, Ariel Bensimon, Ulrich Elling, Alessio Ciulli, Giulio Superti-Furga (Lead / Corresponding author)

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Biochemistry, Genetics and Molecular Biology