@article{2bcd8dff53534294a64acfe1c22e7847,
title = "The identification a novel, selective, non-steroidal, functional glucocorticoid receptor antagonist",
abstract = "The identification of novel, potent, non-steroidal/small molecule functional GR antagonist GSK1564023A selective over PR is described. Associated structure-activity relationships and the process of optimisation of an initial HTS hit are also described.",
author = "Joseph Rimland and Angela Dunne and Hunjan, {Suchete S} and Rosemary Sasse and Iain Uings and Dino Montanari and Matilde Caivano and Poonam Shah and David Standing and David Gray and David Brown and William Cairns and Ryan Trump and Smith, {Paul W} and Nicolas Bertheleme and Pier D'Alessandro and Sheraz Gul and Mythily Vimal and Smith, {David N} and Watson, {Stephen P}",
note = "2010 Elsevier Ltd. All rights reserved.",
year = "2010",
month = apr,
doi = "10.1016/j.bmcl.2010.01.133",
language = "English",
volume = "20",
pages = "2340--3",
journal = "Bioorganic & Medicinal Chemistry Letters",
issn = "1464-3405",
publisher = "Elsevier",
number = "7",
}