Through the "gatekeeper door": exploiting the active kinase conformation

Fabio Zuccotto; Elena Ardini; Elena Casale; Mauro Angiolini

doi:10.1021/jm901443h

Through the "gatekeeper door": exploiting the active kinase conformation

Fabio Zuccotto (Lead / Corresponding author), Elena Ardini, Elena Casale, Mauro Angiolini

Drug Discovery Unit

Research output: Contribution to journal › Review article › peer-review

336 Citations (Scopus)

Original language	English
Pages (from-to)	2681-2694
Number of pages	14
Journal	Journal of Medicinal Chemistry
Volume	53
Issue number	7
Early online date	14 Dec 2009
DOIs	https://doi.org/10.1021/jm901443h
Publication status	Published - 8 Apr 2010

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AU - Casale, Elena

AU - Angiolini, Mauro

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Through the "gatekeeper door": exploiting the active kinase conformation

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