Through the "gatekeeper door": exploiting the active kinase conformation

Fabio Zuccotto; Elena Ardini; Elena Casale; Mauro Angiolini

doi:10.1021/jm901443h

Through the "gatekeeper door": exploiting the active kinase conformation

Fabio Zuccotto (Lead / Corresponding author), Elena Ardini, Elena Casale, Mauro Angiolini

Drug Discovery Unit

Research output: Contribution to journal › Review article

302 Citations (Scopus)

Original language	English
Pages (from-to)	2681-2694
Number of pages	14
Journal	Journal of Medicinal Chemistry
Volume	53
Issue number	7
Early online date	14 Dec 2009
DOIs	https://doi.org/10.1021/jm901443h
Publication status	Published - 8 Apr 2010

Cite this

Zuccotto, F., Ardini, E., Casale, E., & Angiolini, M. (2010). Through the "gatekeeper door": exploiting the active kinase conformation. Journal of Medicinal Chemistry, 53(7), 2681-2694. https://doi.org/10.1021/jm901443h

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Access to Document

10.1021/jm901443h

Link to publication in Scopus