Through the "gatekeeper door": exploiting the active kinase conformation

Fabio Zuccotto; Elena Ardini; Elena Casale; Mauro Angiolini

doi:10.1021/jm901443h

Through the "gatekeeper door": exploiting the active kinase conformation

Fabio Zuccotto (Lead / Corresponding author), Elena Ardini, Elena Casale, Mauro Angiolini

Drug Discovery Unit

Research output: Contribution to journal › Review article › peer-review

458 Citations (Scopus)

Original language	English
Pages (from-to)	2681-2694
Number of pages	14
Journal	Journal of Medicinal Chemistry
Volume	53
Issue number	7
Early online date	14 Dec 2009
DOIs	https://doi.org/10.1021/jm901443h
Publication status	Published - 8 Apr 2010

ASJC Scopus subject areas

Molecular Medicine
Drug Discovery

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10.1021/jm901443h

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title = "Through the {"}gatekeeper door{"}: exploiting the active kinase conformation",

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T2 - exploiting the active kinase conformation

AU - Zuccotto, Fabio

AU - Ardini, Elena

AU - Casale, Elena

AU - Angiolini, Mauro

PY - 2010/4/8

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JO - Journal of Medicinal Chemistry

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Through the "gatekeeper door": exploiting the active kinase conformation

ASJC Scopus subject areas

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