Through the "gatekeeper door": exploiting the active kinase conformation

Fabio Zuccotto; Elena Ardini; Elena Casale; Mauro Angiolini

doi:10.1021/jm901443h

Through the "gatekeeper door": exploiting the active kinase conformation

Fabio Zuccotto (Lead / Corresponding author)
, Elena Ardini
, Elena Casale
, Mauro Angiolini

Drug Discovery Unit

Research output: Contribution to journal › Review article › peer-review

479 Citations (Scopus)

Original language	English
Pages (from-to)	2681-2694
Number of pages	14
Journal	Journal of Medicinal Chemistry
Volume	53
Issue number	7
Early online date	14 Dec 2009
DOIs	https://doi.org/10.1021/jm901443h
Publication status	Published - 8 Apr 2010

ASJC Scopus subject areas

Molecular Medicine
Drug Discovery

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10.1021/jm901443h

Cite this

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title = "Through the {"}gatekeeper door{"}: exploiting the active kinase conformation",

author = "Fabio Zuccotto and Elena Ardini and Elena Casale and Mauro Angiolini",

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journal = "Journal of Medicinal Chemistry",

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TY - JOUR

T1 - Through the "gatekeeper door"

T2 - exploiting the active kinase conformation

AU - Zuccotto, Fabio

AU - Ardini, Elena

AU - Casale, Elena

AU - Angiolini, Mauro

PY - 2010/4/8

Y1 - 2010/4/8

UR - https://www.scopus.com/pages/publications/77950573400

U2 - 10.1021/jm901443h

DO - 10.1021/jm901443h

M3 - Review article

C2 - 20000735

AN - SCOPUS:77950573400

SN - 0022-2623

VL - 53

SP - 2681

EP - 2694

JO - Journal of Medicinal Chemistry

JF - Journal of Medicinal Chemistry

IS - 7

ER -

Through the "gatekeeper door": exploiting the active kinase conformation

ASJC Scopus subject areas

Access to Document

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